Clinical Pipeline and Drug
Discovery Collaborations

Astex Pharmaceuticals™ has established a broad pipeline of small molecule, molecularly targeted drugs using its drug discovery engine, Pyramid™. Pyramid™ is also used to support the Company’s drug discovery collaborations with leading pharmaceutical company partners.

Clinical Pipeline

Program

Phase 1

Phase 2

Phase 3

Marketed

Partner

Novartis *
*Option to license.

Drug Discovery Collaborations

Program

Discovery

Preclinical

Phase 1

Phase 2

Partner

Discovery Obligations Completed

Candidate Selected
Janssen

Discovery Obligations Ongoing

Progress confidential
gsk
Progress confidential
Janssen
†Pending.