Woodhead et al. “Discovery of (2,4-Dihydroxy-5-isopropylphenyl)-[5-(4-methylpiperazin-1-ylmethyl)-1,3-dihydroisoindol-2-yl]methanone (AT13387), a Novel Inhibitor of the Molecular Chaperone Hsp90 by Fragment Based Drug Design.” Journal of Medicinal Chemistry 53, no. 16 2010: 5956–5969. DOI: 10.1021/jm100060b.

Woodhead et al. “Discovery of (2,4-Dihydroxy-5-isopropylphenyl)-[5-(4-methylpiperazin-1-ylmethyl)-1,3-dihydroisoindol-2-yl]methanone (AT13387), a Novel Inhibitor of the Molecular Chaperone Hsp90 by Fragment Based Drug Design.” Journal of Medicinal Chemistry 53, no. 16 2010: 5956–5969. DOI: 10.1021/jm100060b.